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Aerospatiale Puma, Super Puma, & Cougar
Aerospatiale Puma, Super Puma, & Cougar
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Aerospatiale Puma, Super Puma, & Cougar
Structure-Based Discovery of 4-(6-Methoxy-2-methyl-4-(quinolin-4-yl)-9H-pyrimido[4,5-b]indol-7-yl)-3,5-dimethylisoxazole (CD161) as a Potent and Orally Bioavailable BET Bromodomain Inhibitor | Journal of Medicinal Chemistry